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AC5216 CAS 226954-04-7

AC5216 CAS 226954-04-7

In Intermediates, Pharmaceutical Chemicals, Products

Name

AC5216

Synonyms

EMapunil;XBD-173;N-Benzyl-N-ethyl-2-(7-Methyl-8-oxo-2-phenyl-7,8-dihydro-9H-purin-9-yl)acetaMide;9H-Purine-9-acetaMide,N-ethyl-7,8-dihydro-7-Methyl-8-oxo-2-phenyl-N-(phenylMethyl)-;AC 5216 (Emapunil);N-Ethyl-7,8-dihydro-7-methyl-8-oxo-2-phenyl-N-(phenylmethyl)-9H-purine-9-acetamide

Molecular Formula

C23H23N5O2

Molecular Weight

401.46

CAS Number (Or Watson Number for Non-CAS Products)

226954-04-7

EINECS

Specs/Standards

98%min

Use

Emapunil (AC-5216, XBD-173) is an anxiolytic drug which acts as a selective agonist at the peripheral benzodiazepine receptor, also known as the mitochondrial 18 kDa translocator protein or TSPO. This protein has multiple functions, among which is regulation of steroidogenesis, particularly the production of neuroactive steroids such as allopregnanolone in the brain. In both animal and human trials, emapunil produced fast acting anxiolytic and anti-panic effects, without producing sedation or withdrawal symptoms following cessation of use.Emapunil is also used in its 11C radiolabelled form to map the distribution of TSPO receptors in the brain.

Sales Link

This product is exclusively sold through our sales company Watson International Ltd and please refer to the link below for inquiries
http://watson-int.com/AC5216-cas-226954-04-7/